Chemistry:Azapride

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Short description: Chemical compound
Azapride
Azapride.png
Clinical data
Other namesAzidoclebopride
ATC code
  • None
Identifiers
CAS Number
PubChem CID
ChemSpider
UNII
Chemical and physical data
FormulaC20H22ClN5O2
Molar mass399.88 g·mol−1
3D model (JSmol)
  (verify)

Azapride is the azide derivative of the dopamine antagonist clebopride synthesized in order to label dopamine receptors.[1][2] It is an irreversible dopamine antagonist.[2]

References

  1. "A photoaffinity ligand for dopamine D2 receptors: azidoclebopride". Molecular Pharmacology 27 (2): 193–9. February 1985. PMID 3969068. 
  2. 2.0 2.1 "Photoaffinity labelling of dopamine receptors. Synthesis and binding characteristics of azapride". European Journal of Biochemistry 145 (2): 273–8. December 1984. doi:10.1111/j.1432-1033.1984.tb08548.x. PMID 6548707.