Chemistry:MRS7292
From HandWiki
MRS7292 is an experimental drug that selectively activates the adenosine A3 receptor with moderate affinity and also inhibits a dopamine reuptake. This combination of mechanisms has been observed in the same molecule.[1][2]
See also
- MRS8209
References
- ↑ "Scaffold Repurposing of Nucleosides (Adenosine Receptor Agonists): Enhanced Activity at the Human Dopamine and Norepinephrine Sodium Symporters". Journal of Medicinal Chemistry 60 (7): 3109–3123. April 2017. doi:10.1021/acs.jmedchem.7b00141. PMID 28319392.
- ↑ "Direct Comparison of (N)-Methanocarba and Ribose-Containing 2-Arylalkynyladenosine Derivatives as A3 Receptor Agonists". ACS Medicinal Chemistry Letters 11 (10): 1935–1941. October 2020. doi:10.1021/acsmedchemlett.9b00637. PMID 33062176.
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