Chemistry:Beta-3 adrenergic antagonist

From HandWiki

A Beta-3 adrenergic antagonist3-adrenoceptor antagonist) is an adrenergic antagonist which blocks the Beta-3 adrenergic receptors of cells, with either high specificity (an antagonist which is selective for β3 adrenoceptors) like L-748,328, L-748,337 and SR 59230A or non-specifically (an antagonist for β3 and for β1 or β2 adrenoceptors) like the non-selective betablocker Carvedilol.[1]

See also

References

  1. "Potent and selective human beta(3)-adrenergic receptor antagonists.". The Journal of Pharmacology and Experimental Therapeutics 290 (2): 649–55. Aug 1999. PMID 10411574. http://jpet.aspetjournals.org/content/290/2/649.long.