Chemistry:Azabon
From HandWiki
Short description: Chemical compound
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| Formula | C14H20N2O2S |
| Molar mass | 280.386 |
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Azabon is a central nervous system stimulant of the sulfonamide class[1] that is also used as a nootropic.[2] As it is a sulpha drug, care must be taken during administration, and certain individuals must avoid azabon altogether to prevent an allergic reaction. Despite being a sulfonamide, azabon has poor antibacterial potency, although this decreased activity is common among other benzenesulfonamides with two substituents on N1. Azabon is synthesized from 3-azabicyclo-[2.2.2]nonane, which is itself prepared by pyrolysis of aliphatic diamine.[3]
See also
References
- ↑ Vetter D, Rau H, "Dipeptide-based prodrug linkers for aromatic amine-containing drugs", WO patent 2011089215, published 28 July 2011, assigned to Ascendis Pharma AS
- ↑ "Chemical Structure-Related Drug-Like Criteria of Global Approved Drugs". Molecules 21 (1): 75. January 2016. doi:10.3390/molecules21010075. PMID 26771590.
- ↑ The Organic Chemistry of Drug Synthesis. 2. Wiley Interscience. 1980. p. 115. ISBN 0-471-04392-3. https://www.mobt3ath.com/uplode/book/book-19950.pdf.
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