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Short description
Imidafenacin Clinical data Routes of By mouth ATC code Legal status Legal status
In general: ℞ (Prescription only)
Identifiers
4-(2-methyl-1H -imidazol-1-yl)-2,2-diphenylbutanamide
CAS Number PubChem CID ChemSpider UNII ChEMBL Chemical and physical data Formula C 20 H 21 N 3 O Molar mass −1 3D model (JSmol )
CC1=NC=CN1CCC(C2=CC=CC=C2)(C3=CC=CC=C3)C(=O)N
InChI=1S/C20H21N3O/c1-16-22-13-15-23(16)14-12-20(19(21)24,17-8-4-2-5-9-17)18-10-6-3-7-11-18/h2-11,13,15H,12,14H2,1H3,(H2,21,24)
N Key:SQKXYSGRELMAAU-UHFFFAOYSA-N
N N Y (what is this?) (verify)
Imidafenacin (INN) is a urinary antispasmodic of the anticholinergic class.
Pharmacol:[1]
References
↑ "Effects of imidafenacin (KRP-197/ONO-8025), a new anti-cholinergic agent, on muscarinic acetylcholine receptors. High affinities for M3 and M1 receptor subtypes and selectivity for urinary bladder over salivary gland". Arzneimittelforschung 57 (2): 92–100. 2007. doi :10.1055/s-0031-1296589 . PMID 17396619 .
mAChRs
Agonists Antagonists
3-Quinuclidinyl benzilate 4-DAMP Aclidinium bromide (+formoterol )Abediterol AF-DX 250 AF-DX 384 Ambutonium bromide Anisodamine Anisodine Antihistamines (first-generation) (e.g., brompheniramine , buclizine , captodiame , chlorphenamine (chlorpheniramine) , cinnarizine , clemastine , cyproheptadine , dimenhydrinate , [[Chemistry:Dimetdimetindene, Diphenhydramine |diphenhydramine]], doxylamine , meclizine , mepyramine (pyrilamine) , mequitazine , perlapine , phenindamine , pheniramine , Phenyltoloxamine|Phenyltoloxamine ]]]], promethazine , propiomazine , triprolidine )AQ-RA 741 Atropine Atropine methonitrate Atypical antipsychotics (e.g., clozapine, Chemistry :Fluperlapine
Precursors (and prodrugs)
Original source: https://en.wikipedia.org/wiki/Imidafenacin. Read more
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