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Template:Transient receptor potential channel modulators
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v
t
e
TRP
channel
modulators
TRPA
Activators
4-Hydroxynonenal
4-Oxo-2-nonenal
4,5-EET
12S-HpETE
15-Deoxy-Δ
12,14
-prostaglandin J2
α-Sanshool
(
ginger
,
Sichuan
and
melegueta peppers
)
Acrolein
Allicin
(
garlic
)
Allyl isothiocyanate
(
mustard
,
radish
,
horseradish
,
wasabi
)
AM404
Bradykinin
Cannabichromene
(
cannabis
)
Cannabidiol
(
cannabis
)
Cannabigerol
(
cannabis
)
Cinnamaldehyde
(
cinnamon
)
CR gas (dibenzoxazepine; DBO)
CS gas (2-chlorobenzal malononitrile)
Curcumin
(
turmeric
)
Dehydroligustilide
(
celery
)
Diallyl disulfide
Dicentrine
(
Lindera
spp.)
Farnesyl thiosalicylic acid
Formalin
Gingerols
(
ginger
)
Hepoxilin A3
Hepoxilin B3
Hydrogen peroxide
Icilin
Isothiocyanate
Ligustilide
(
celery
,
Angelica acutiloba
)
Linalool
(
Sichuan pepper
,
thyme
)
Methylglyoxal
Methyl salicylate
(
wintergreen
)
N-Methylmaleimide
Nicotine
(
tobacco
)
Oleocanthal
(
olive oil
)
Paclitaxel
(
Pacific yew
)
Paracetamol (acetaminophen)
PF-4840154
Phenacyl chloride
Polygodial
(
Dorrigo pepper
)
Shogaols
(
ginger
,
Sichuan
and
melegueta peppers
)
Tear gases
Tetrahydrocannabinol
(
cannabis)
Thiopropanal S-oxide
(
onion
)
Umbellulone
(
Umbellularia californica
)
WIN 55,212-2
Blockers
Dehydroligustilide
(
celery
)
Nicotine
(
tobacco
)
Ruthenium red
TRPC
Activators
Adhyperforin
(
St John's wort
)
Diacyl glycerol
GSK1702934A
Hyperforin
(
St John's wort
)
Substance P
Blockers
DCDPC
DHEA-S
Flufenamic acid
GSK417651A
GSK2293017A
Meclofenamic acid
N-(p-Amylcinnamoyl)anthranilic acid
Niflumic acid
Pregnenolone sulfate
Progesterone
Pyr3
Tolfenamic acid
TRPM
Activators
ADP-ribose
BCTC
Calcium
(intracellular)
Cold
Coolact P
Cooling Agent 10
CPS-369
Eucalyptol
(
eucalyptus
)
Frescolat MGA
Frescolat ML
Geraniol
Hydroxycitronellal
Icilin
Linalool
Menthol
(
mint
)
PMD 38
Pregnenolone sulfate
Rutamarin
(
Ruta graveolens
)
Steviol glycosides
(e.g.,
stevioside
) (
Stevia rebaudiana
)
Sweet
tastants
(e.g.,
glucose
,
fructose
,
sucrose
; indirectly)
Thio-BCTC
WS-3
WS-12
WS-23
Blockers
Capsazepine
Clotrimazole
DCDPC
Elismetrep
Flufenamic acid
Meclofenamic acid
Mefenamic acid
N-(p-Amylcinnamoyl)anthranilic acid
Nicotine
(
tobacco
)
Niflumic acid
Ruthenium red
Rutamarin
(
Ruta graveolens
)
Tolfenamic acid
TPPO
TRPML
Activators
MK6-83
PI(3,5)P
2
SF-22
TRPP
Activators
Triptolide
(
Tripterygium wilfordii
)
Blockers
Ruthenium red
TRPV
Activators
2-APB
5',6'-EET
9-HODE
9-oxoODE
12S-HETE
12S-HpETE
13-HODE
13-oxoODE
20-HETE
α-Sanshool
(
ginger
,
Sichuan
and
melegueta peppers
)
Allicin
(
garlic
)
AM404
Anandamide
Bisandrographolide
(
Andrographis paniculata
)
Camphor
(
camphor laurel
,
rosemary
,
camphorweed
,
African blue basil
,
camphor basil)<
!--TRPV1 and TRPV3-->
Cannabidiol
(
cannabis
)
Cannabidivarin
(
cannabis
)
Capsaicin
(
chili pepper
)
Carvacrol
(
oregano
,
thyme
,
pepperwort,
wild bergamot,
others)
DHEA
Diacyl glycerol
Dihydrocapsaicin
(
chili pepper
)
Estradiol
Eugenol
(
basil
,
clove
)
Evodiamine
(
Euodia ruticarpa
)
Gingerols
(
ginger
)
GSK1016790A
Heat
Hepoxilin A3
Hepoxilin B3
Homocapsaicin
(
chili pepper
)
Homodihydrocapsaicin
(
chili pepper
)
Incensole
(
incense
)
Lysophosphatidic acid
Low
pH
(acidic conditions)
Menthol
(
mint
)
N-Arachidonoyl dopamine
N-Oleoyldopamine
N-Oleoylethanolamide
Nonivamide (PAVA)
(
PAVA spray
)
Nordihydrocapsaicin
(
chili pepper
)
Paclitaxel
(
Pacific yew
)
Paracetamol (acetaminophen)
Phorbol esters
(e.g.,
4α-PDD
)
Piperine
(
black pepper
,
long pepper)
Polygodial
(
Dorrigo pepper
)
Probenecid
Protons
RhTx
Rutamarin
(
Ruta graveolens
)
Resiniferatoxin
(RTX) (
Euphorbia resinifera
/
pooissonii
)
Shogaols
(
ginger
,
Sichuan
and
melegueta peppers
)
Tetrahydrocannabivarin
(
cannabis
)
Thymol
(
thyme
,
oregano
)
Tinyatoxin
(
Euphorbia resinifera
/
pooissonii
)
Tramadol
Vanillin
(
vanilla
)
Zucapsaicin
Blockers
α-Spinasterol
(
Vernonia tweediana
)
AMG-517
Asivatrep
BCTC
Cannabigerol
(
cannabis
)
Cannabigerolic acid
(
cannabis
)
Cannabigerovarin
(
cannabis
)
Cannabinol
(
cannabis
)
Capsazepine
DCDPC
DHEA
DHEA-S
Flufenamic acid
GRC-6211
HC-067047
Lanthanum
Mavatrep
Meclofenamic acid
N-(p-Amylcinnamoyl)anthranilic acid
NGD-8243
Niflumic acid
Pregnenolone sulfate
RN-1734
RN-9893
Ruthenium red
SB-705498
Tivanisiran
Tolfenamic acid
See also:
Receptor/signaling modulators
•
Ion channel modulators
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