Chemistry:TRPV3-74a
From HandWiki
Short description: Chemical compound
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| Formula | C17H17F3N2O2 |
| Molar mass | 338.330 g·mol−1 |
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TRPV3-74a is a drug which acts as a selective antagonist for the TRPV3 calcium channel. It has analgesic effects in animal studies against both neuropathic pain and normal pain responses.[1][2]
References
- ↑ "Synthesis and Pharmacology of (Pyridin-2-yl)methanol Derivatives as Novel and Selective Transient Receptor Potential Vanilloid 3 Antagonists". Journal of Medicinal Chemistry 59 (10): 4926–47. May 2016. doi:10.1021/acs.jmedchem.6b00287. PMID 27077528.
- ↑ "Synthesis of a TRPV3 Antagonist.". Synfacts 13 (2): 123. February 2017. doi:10.1055/s-0036-1589889.
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