Chemistry:Timelotem

Short description: Chemical compound

Timelotem

Clinical data
ATC code	none
Identifiers
IUPAC name 10-fluoro-3-methyl-7-thiophen-2-yl-2,4,4a,5-tetrahydro-1H-pyrazino[1,2-a][1,4]benzodiazepine
CAS Number	96306-34-2
PubChem CID	65844
Chemical and physical data
Formula	C17H18FN3S
Molar mass	315.41 g·mol−1
3D model (JSmol)	Interactive image
SMILES CN1CCN2C(C1)CN=C(C3=C2C=C(C=C3)F)C4=CC=CS4
InChI InChI=1S/C17H18FN3S/c1-20-6-7-21-13(11-20)10-19-17(16-3-2-8-22-16)14-5-4-12(18)9-15(14)21/h2-5,8-9,13H,6-7,10-11H2,1H3 Key:ICHHTOMWWAMJQP-UHFFFAOYSA-N

Timelotem is a benzodiazepine derivative with an unusual activity profile. Unlike most benzodiazepines, timelotem has little or no activity at the GABA_A receptor, but instead acts as an atypical antipsychotic drug with similar pharmacology and effects to the structurally related drug clozapine. It has two enantiomers, but has only been studied as the racemic mix.

See also

• Olanzapine