Chemistry:ADRIANA
From HandWiki
ADRIANA is a selective α2B-adrenergic receptor antagonist.[1] It is described as highly selective over the α2A- and α2C-adrenergic receptors.[1] The drug stimulates norepinephrine release in the spinal dorsal horn and has potent analgesic effects in rodents and non-human primates.[1] It is orally active.[1] ADRIANA was first described in the scientific literature by Masayasu Toyomoto and colleagues in 2025.[1] It is said to be the first selective α2B-adrenergic receptor antagonist to have been developed.[1]
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