Chemistry:RU-57073
From HandWiki
Short description: Chemical compound
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| Drug class | Nonsteroidal antiandrogen |
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| Formula | C15H14F3N3O2S |
| Molar mass | 357.35 g·mol−1 |
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RU-57073 is a nonsteroidal antiandrogen which was never marketed.[1][2][3] It shows 163% of the affinity of testosterone for the androgen receptor and negligible affinity for other steroid hormone receptors.[1][2]
See also
References
- ↑ 1.0 1.1 "Androgen receptor antagonists (antiandrogens): structure-activity relationships". Curr. Med. Chem. 7 (2): 211–47. February 2000. doi:10.2174/0929867003375371. PMID 10637363.
- ↑ 2.0 2.1 "Non-steroidal antiandrogens: synthesis and biological profile of high-affinity ligands for the androgen receptor". J. Steroid Biochem. Mol. Biol. 48 (1): 111–9. January 1994. doi:10.1016/0960-0760(94)90257-7. PMID 8136296.
- ↑ "RU 58841-myristate--prodrug development for topical treatment of acne and androgenetic alopecia". Pharmazie 60 (1): 8–12. January 2005. PMID 15700772. https://www.ingentaconnect.com/content/govi/pharmaz/2005/00000060/00000001/art00002.
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