Chemistry:GR-45809

From HandWiki

GR-45809 is a kappa opioid receptor (KOR) agonist with use in the treatment of pain.[1][2] It was developed over 30 years ago. It has a structure that is similar to ZT-52656A.

References

  1. ↑ "(2S)-1-(arylacetyl)-2-(aminomethyl)piperidine derivatives: novel, highly selective kappa opioid analgesics". Journal of Medicinal Chemistry 34 (1): 397–403. January 1991. doi:10.1021/jm00105a061. PMID 1846921. 
  2. ↑ "New kappa-receptor agonists based upon a 2-[(alkylamino)methyl]piperidine nucleus". Journal of Medicinal Chemistry 35 (3): 490–501. February 1992. doi:10.1021/jm00081a009. PMID 1310743. 



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