Chemistry:Eptazocine
From HandWiki
Short description: Opioid analgesic
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| Routes of administration | Oral |
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| Formula | C15H21NO |
| Molar mass | 231.339 g·mol−1 |
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Eptazocine (Sedapain) is an opioid analgesic which was introduced in Japan by Morishita in 1987.[1][2][3][4] It acts as a mixed κ-opioid receptor agonist and μ-opioid receptor antagonist.[4][5][6]
See also
- Benzomorphan
References
- ↑ Index nominum 2000: international drug directory. Taylor & Francis US. 2000. p. 396. ISBN 978-3-88763-075-1. https://books.google.com/books?id=5GpcTQD_L2oC&pg=PA396. Retrieved 29 November 2011.
- ↑ American Chemical Society. Division of Medicinal Chemistry (1990). "Cumulative NCE Introduction index, 1983-189, by Indication". Annual Reports in Medicinal Chemistry. Academic Press. p. 381. ISBN 978-0-12-040525-1. https://books.google.com/books?id=NZZbEkldeJAC&pg=PA381. Retrieved 29 November 2011.
- ↑ "The interaction of eptazocine, a novel analgesic, with opioid receptors". Research Communications in Chemical Pathology and Pharmacology 48 (2): 173–181. May 1985. PMID 2992058.
- ↑ 4.0 4.1 "Synthesis of Novel Basic Skeletons Derived from Naltrexone". Chemistry of Opioids. Springer. 21 January 2011. p. 280. ISBN 978-3-642-18106-1. https://books.google.com/books?id=5GUn9E-9irMC&pg=PA280. Retrieved 29 November 2011.
- ↑ "[Preferential action of eptazocine, a novel analgesic, with opioid receptors in isolated guinea pig ileum and mouse vas deferens preparations]" (in ja). Nihon Yakurigaku Zasshi. Folia Pharmacologica Japonica 95 (1): 41–46. January 1990. doi:10.1254/fpj.95.1_41. PMID 2154395.
- ↑ Concise dictionary of pharmacological agents: properties and synonyms. Springer. 1999. p. 113. ISBN 978-0-7514-0499-9. https://books.google.com/books?id=mqaOMOtk61IC&pg=PA113. Retrieved 29 November 2011.
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