Chemistry:Proheptazine
From HandWiki
Short description: Opioid analgesic drug
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| Formula | C17H25NO2 |
| Molar mass | 275.392 g·mol−1 |
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Proheptazine is an opioid analgesic related to pethidine. It was invented in the 1960s.[1]
Proheptazine produces similar effects to other opioids, including analgesia, sedation, euphoria, dizziness and nausea.
In the United States it is a Schedule I Narcotic controlled substance with an ACSCN of 9643 and a 2013 annual aggregate manufacturing quota of zero. The salts in use are the citrate (free base conversion ratio 0.589), hydrobromide (0.773), and hydrochloride (0.883).[2][3]
References
- ↑ "Synthesis and Properties of the Analgesic DL-α-1,3-dimethyl-4-phenyl-4-propionoxyazacycloheptane (Proheptazine).". Journal of Medicinal Chemistry 7: 57–60. January 1964. doi:10.1021/jm00331a013. PMID 14186026.
- ↑ "Quotas - 2014". Diversion Control Division. Drug Enforcement Agency, U.S. Department of Justice. http://www.deadiversion.usdoj.gov/fed_regs/quotas/2014/fr0825.htm.
- ↑ "Conversion Factors for Controlled Substances". Diversion Control Division. Drug Enforcement Agency, U.S. Department of Justice. http://www.deadiversion.usdoj.gov/quotas/conv_factor/index.html.
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