Chemistry:Diampromide
From HandWiki
Short description: Opioid analgesic drug
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| Other names | Diampromide |
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| Formula | C21H28N2O |
| Molar mass | 324.468 g·mol−1 |
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Diampromide is an opioid analgesic from the ampromide family of drugs, related to other drugs such as propiram and phenampromide. It was invented in the 1960s by American Cyanamid,[1] and can be described as a ring-opened analogue of fentanyl.[2]
Diampromide produces similar effects to other opioids, including analgesia, sedation, dizziness and nausea, and is around the same potency as morphine.[3]
Diampromide is in Schedule I of the Controlled Substances Act 1970 of the United States as a Narcotic with ACSCN 9615 with a zero aggregate manufacturing quota as of 2014.[4] It is listed under the Single Convention for the Control of Narcotic Substances 1961 and is controlled in most countries in the same fashion as is morphine.
See also
References
- ↑ "Diphenylalkylenediamines and Methods of Preparation of the Same" US patent 2944081
- ↑ "Theoretical Study of Acyclic FENTANYL ANALOGS With Analgesic Activity: Diampromide and seco-Fentanyl". http://www.ch.ic.ac.uk/ectoc/echet98/pub/028/index.htm.
- ↑ "The synthesis and pharmacological evaluation of 2,3-seco-fentanyl analogues". Journal of the Serbian Chemical Society 69 (11): 955–968. 2004. doi:10.2298/JSC0411955I.
- ↑ "Final Adjusted Aggregate Production Quotas for Schedule I and II Controlled Substances and Assessment of Annual Needs for the List I Chemicals Ephedrine, Pseudoephedrine, and Phenylpropanolamine for 2014". Drug Enforcement Administration. http://www.deadiversion.usdoj.gov/fed_regs/quotas/2014/fr0825.htm.
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