Chemistry:RS-56812

RS-56812
Identifiers
	IUPAC name N-[(3R)-1-azabicyclo[2.2.2]oct-3-yl]-2-(1-methyl-1H-indol-3-yl)-2-oxoacetamide;
CAS Number	143137-35-3;
PubChem CID	6604789;
Chemical and physical data
Formula	C18H21N3O2
Molar mass	311.385 g·mol−1
3D model (JSmol)	Interactive image;
	SMILES c14ccccc4n(C)cc1C(=O)C(=O)NC2CN3CCC2CC3;
	(verify)

Short description: Chemical compound

RS-56812 is a potent and selective partial agonist at the 5HT₃ receptor.^[1] It has been shown to improve performance on animal tests of memory. Its use in humans is not well documented. ^[2]

References

↑ "RS-056812-198: partial agonist on native and antagonist on cloned 5-HT3 receptors". European Journal of Pharmacology 322 (2–3): 229–33. March 1997. doi:10.1016/s0014-2999(96)00993-4. PMID 9098692.
↑ "The 5-HT3 receptor antagonist, RS-56812, enhances delayed matching performance in monkeys". NeuroReport 8 (1): 49–54. December 1996. doi:10.1097/00001756-199612200-00011. PMID 9051751.

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[1] "RS-056812-198: partial agonist on native and antagonist on cloned 5-HT3 receptors". European Journal of Pharmacology 322 (2–3): 229–33. March 1997. doi:10.1016/s0014-2999(96)00993-4. PMID 9098692.

[2] "The 5-HT3 receptor antagonist, RS-56812, enhances delayed matching performance in monkeys". NeuroReport 8 (1): 49–54. December 1996. doi:10.1097/00001756-199612200-00011. PMID 9051751.

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Identifiers

IUPAC name N-[(3R)-1-azabicyclo[2.2.2]oct-3-yl]-2-(1-methyl-1H-indol-3-yl)-2-oxoacetamide
CAS Number	143137-35-3
PubChem CID	6604789
Chemical and physical data
Formula	C₁₈H₂₁N₃O₂
Molar mass	311.385 g·mol⁻¹
3D model (JSmol)	Interactive image
SMILES c14ccccc4n(C)cc1C(=O)C(=O)NC2CN3CCC2CC3
(verify)

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