Chemistry:CUMYL-THPINACA
From HandWiki
Short description: Chemical compound
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| Formula | C23H27N3O2 |
| Molar mass | 377.488 g·mol−1 |
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CUMYL-THPINACA (also known as SGT-42) is an indazole-3-carboxamide based synthetic cannabinoid.[1][2] CUMYL-THPINACA acts as a potent agonist for the cannabinoid receptors, with approximately 6x selectivity for CB1, having an EC50 of 0.1nM for human CB1 receptors and 0.59nM for human CB2 receptors.[3]
Legal status
Sweden's public health agency suggested to classify CUMYL-THPINACA as hazardous substance on November 10, 2014.[4]
As of October 2015 CUMYL-THPINACA is a controlled substance in China.[5]
See also
- 5F-CUMYL-PINACA
- 5F-SDB-006
- ADAMANTYL-THPINACA
- CUMYL-4CN-BINACA
- CUMYL-CBMINACA
- CUMYL-PICA
- CUMYL-PINACA
- SDB-006
- NNE1
References
- ↑ "CUMYL-THPINACA". Cayman Chemical. https://www.caymanchem.com/app/template/Product.vm/catalog/17210.
- ↑ "Phase I In Vitro Metabolic Profiling of the Synthetic Cannabinoid Receptor Agonists CUMYL-THPINACA and ADAMANTYL-THPINACA". Metabolites 11 (8): 470. July 2021. doi:10.3390/metabo11080470. PMID 34436411.
- ↑ Bowden MJ, Williamson JP, "Cannabinoid compounds", WO patent 2014167530, published 2014-10-16
- ↑ "Cannabinoider föreslås bli klassade som hälsofarlig vara". http://www.folkhalsomyndigheten.se/nyheter-och-press/nyhetsarkiv/2014/november/cannabinoider-foreslas-bli-klassade-som-halsofarlig-vara/.
- ↑ "关于印发《非药用类麻醉药品和精神药品列管办法》的通知" (in zh). China Food and Drug Administration. 27 September 2015. http://www.sfda.gov.cn/WS01/CL0056/130753.html.
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