Chemistry:Fasiplon
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Short description: Chemical compound
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| Formula | C13H15N5O2 |
| Molar mass | 273.296 g·mol−1 |
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Fasiplon binds strongly to benzodiazepine sites on the GABAA receptor and has similar anxiolytic effects in animals, but with less sedative or muscle relaxant action.[1] It was developed by a team at Roussel Uclaf in the 1990s[2]
References
- ↑ "2-(oxadiazolyl)- and 2-(thiazolyl)imidazo[1,2-a]pyrimidines as agonists and inverse agonists at benzodiazepine receptors". Journal of Medicinal Chemistry 34 (7): 2060–7. July 1991. doi:10.1021/jm00111a021. PMID 1648620.
- ↑ US Patent 5869481 Anticonvulsive 1-ar(alk)ylimidazolin-2-ones and process for making
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