Chemistry:Ciclotizolam
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Short description: Chemical compound
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Formula | C20H18BrClN4S |
Molar mass | 461.81 g·mol−1 |
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Ciclotizolam[1] (WE-973) is a drug which is a thienotriazolodiazepine derivative. It is a partial agonist for the benzodiazepine site of the GABAA receptor, with similar binding affinity to related compounds like brotizolam, but a low efficacy.[2][3]
See also
References
- ↑ DE Patent 2445430
- ↑ "Pharmacological and neurochemical properties of 1,4-diazepines with two annelated heterocycles ('hetrazepines')". European Journal of Pharmacology 109 (1): 19–31. February 1985. doi:10.1016/0014-2999(85)90535-7. PMID 2986988.
- ↑ "Relative efficacies of 1,4-diazepines on GABA-stimulated chloride influx in rat brain vesicles". Life Sciences 45 (4): 349–58. 1989. doi:10.1016/0024-3205(89)90145-8. PMID 2569655.
Original source: https://en.wikipedia.org/wiki/Ciclotizolam.
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