Chemistry:Pipradimadol

From HandWiki

Pipradimadol (FU 29-245) is an analgesic, antiserotoninergic agent and potentially an antidepressant.[1][2] The pharmacology is said to be mediated through the opiate receptor. The potency is on the same order of magnitude as for morphine.[3]

See also

  • Pipramadol

References

  1. "Synthesis and pharmacological studies of 4,4-disubstituted piperidines: a new class of compounds with potent analgesic properties". Journal of Medicinal Chemistry 26 (1): 42–50. January 1983. doi:10.1021/jm00355a010. PMID 6600791. 
  2. "Human EEG slow-wave sleep increased by a serotonin antagonist". Electroencephalography and Clinical Neurophysiology 54 (5): 583–6. November 1982. doi:10.1016/0013-4694(82)90044-x. PMID 6181982. 
  3. Rissi E, Ebnother A, "(4-Hydroxy-4-piperidyl)-alkanoic acid amides", US patent 4178377, issued 11 December 1979.