Chemistry:Revospirone

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Short description: Chemical compound
Revospirone
Revospirone.svg
Clinical data
ATC code
  • none
Identifiers
CAS Number
PubChem CID
ChemSpider
UNII
Chemical and physical data
FormulaC18H21N5O3S
Molar mass387.46 g·mol−1

Revospirone (Bay Vq 7813) is an azapirone drug which was patented as a veterinary tranquilizer but was never marketed.[1] It acts as a selective 5-HT1A receptor partial agonist.[2] Similarly to other azapirones such as buspirone, revospirone produces 1-(2-pyrimidinyl)piperazine (1-PP) as an active metabolite.[2] As a result, it also acts as an α2-adrenergic receptor antagonist to an extent.[2]

References

  1. ↑ Dictionary of Pharmacological Agents. CRC Press. 1997. p. 1744. ISBN 978-0-412-46630-4. https://books.google.com/books?id=A0THacd46ZsC&pg=PA1744. Retrieved 13 May 2012. 
  2. ↑ 2.0 2.1 2.2 "The behavioural responses to 8-OH-DPAT, ipsapirone and the novel 5-HT1A receptor agonist Bay Vq 7813 in the pig". Naunyn-Schmiedeberg's Archives of Pharmacology 342 (3): 271–7. September 1990. doi:10.1007/bf00169437. PMID 2149168. 




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